Discovery of Low Nanomolar and Subnanomolar Inhibitors of the Mycobacterial β-Carbonic Anhydrases Rv1284 and Rv3273-Reference-Cited by-同舟云学术

Discovery of Low Nanomolar and Subnanomolar Inhibitors of the Mycobacterial β-Carbonic Anhydrases Rv1284 and Rv3273

Published:2009-05-13 Issue:13 Volume:52 Page:4063-4067
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Güzel Özlen¹,Maresca Alfonso¹,Scozzafava Andrea¹,Salman Aydın¹,Balaban Alexandru T.¹,Supuran Claudiu T.¹

Affiliation:

1. Istanbul University, Faculty of Pharmacy, Department of Pharmaceutical Chemistry, 34116 Beyazıt, Istanbul, Turkey, Università degli Studi di Firenze, Polo Scientifico, Laboratorio di Chimica Bioinorganica, Rm. 188, Via della Lastruccia 3, 50019 Sesto Fiorentino (Florence), Italy, Texas A&M University at Galveston, 5007 Avenue U, Galveston, Texas 77551

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm9004016

Reference33 articles.

1. Molecular Cloning, Characterization, and Inhibition Studies of the Rv1284 β-Carbonic Anhydrase from Mycobacterium tuberculosis with Sulfonamides and a Sulfamate

2. Carbonic Anhydrase Inhibitors. Cloning, Characterization, and Inhibition Studies of a New β-Carbonic Anhydrase from Mycobacterium tuberculosis

3. Structure and Function of Carbonic Anhydrases from Mycobacterium tuberculosis

4. Structural Mechanics of the pH-dependent Activity of β-Carbonic Anhydrase from Mycobacterium tuberculosis

5. Deciphering the biology of Mycobacterium tuberculosis from the complete genome sequence

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