Allosteric Competitive Inhibitors of the Glucose-1-phosphate Thymidylyltransferase (RmlA) from Pseudomonas aeruginosa

Author:

Alphey Magnus S.1,Pirrie Lisa12,Torrie Leah S.3,Boulkeroua Wassila Abdelli1,Gardiner Mary3,Sarkar Aurijit3,Maringer Marko4,Oehlmann Wulf5,Brenk Ruth3,Scherman Michael S.6,McNeil Michael6,Rejzek Martin7,Field Robert A.7,Singh Mahavir5,Gray David3,Westwood Nicholas J.12,Naismith James H.1

Affiliation:

1. Biomedical Sciences Research Complex, University of St. Andrews, St. Andrews KY16 9ST, U.K.

2. School of Chemistry, University of St. Andrews and EaStCHEM, St. Andrews KY16 9ST, U.K.

3. Biological Chemistry and Drug Discovery, College of Life Sciences, University of Dundee, Dundee DD1 5EH, U.K.

4. mfd Diagnostics GmbH, Mikroforum Ring 5, 55234 Wendelsheim, Germany

5. Lionex GmbH, Salzdahlumer Str. 196, 38126 Braunschweig, Germany

6. Department of Microbiology, Immunology and Pathology, Colorado State University, 1682 Campus Delivery, Ft. Collins, Colorado 80523-1682, United States

7. Department of Biological Chemistry, John Innes Centre, Norwich NR4 7UH, U.K.

Publisher

American Chemical Society (ACS)

Subject

Molecular Medicine,General Medicine,Biochemistry

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