Synthesis of Differentially Protected Azatryptophan Analogs via Pd2(dba)3/XPhos Catalyzed Negishi Coupling of N-Ts Azaindole Halides with Zinc Derivative from Fmoc-Protected tert-Butyl (R)-2-Amino-3-iodopropanoate-Reference-Cited by-同舟云学术

Synthesis of Differentially Protected Azatryptophan Analogs via Pd2(dba)3/XPhos Catalyzed Negishi Coupling of N-Ts Azaindole Halides with Zinc Derivative from Fmoc-Protected tert-Butyl (R)-2-Amino-3-iodopropanoate

Published:2020-08-10 Issue:17 Volume:85 Page:11519-11530
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

Nimje Roshan Y¹,Vytla Devaiah¹,Kuppusamy Prakasam¹,Velayuthaperumal Rajeswari¹,Jarugu Lokesh Babu¹,Reddy China Anki¹,Chikkananjaiah Nanjundaswamy Kanikahalli¹,Rampulla Richard A.²,Cavallaro Cullen L.²,Li Jianqing³^ORCID,Mathur Arvind²,Gupta Anuradha¹^ORCID,Roy Amrita¹^ORCID

Affiliation:

1. Department of Discovery Synthesis, Biocon Bristol-Myers Squibb R&D Center, Syngene International Ltd., Biocon Park, Plot No. 2 and 3, Bommasandra-Jigani Road, Bangalore-560 100, India

2. Small Molecule Drug Discovery, Bristol-Myers Squibb Research and Development, P.O. Box 5400, Princeton, New Jersey 08543-4000, United States

3. Small Molecule Drug Discovery, Bristol-Myers Squibb Research and Development, 100 Binney Street, Cambridge, Massachusetts 02142, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.joc.0c00973

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