Palladium-Catalyzed Regioselective Alkynylation of Pyrroles and Azoles under Mild Conditions: Application to the Synthesis of a Dopamine D-4 Receptor Agonist-Reference-Cited by-同舟云学术

Palladium-Catalyzed Regioselective Alkynylation of Pyrroles and Azoles under Mild Conditions: Application to the Synthesis of a Dopamine D-4 Receptor Agonist

Published:2015-07-24 Issue:15 Volume:80 Page:7519-7529
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

Brachet Etienne¹²,Belmont Philippe¹²

Affiliation:

1. Université Paris Descartes, Faculté de Pharmacie de Paris, UMR CNRS 8638 (COMETE), 4 avenue de l’Observatoire, Paris FR-75006, France

2. Université Sorbonne Paris Cité (USPC), 12 rue de l’école de Médecine, Paris FR-75006, France

Funder

Institut National Du Cancer

Centre National de la Recherche Scientifique

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.joc.5b01093

Reference54 articles.

1. The Combinatorial Synthesis of Bicyclic Privileged Structures or Privileged Substructures

2. Synthesis of Oxygen- and Nitrogen-Containing Heterocycles by Ring-Closing Metathesis

3. From Nature to Drug Discovery: The Indole Scaffold as a ‘Privileged Structure’

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