Cyclization of Methyl-Coumalate-Derived Methyl 1-Benzamido-6-oxo-1,6-dihydropyridine-3-carboxylates: Assembly of the [1,2,4]Triazolo[1,5-a]pyridine Ring System-Reference-Cited by-同舟云学术

Cyclization of Methyl-Coumalate-Derived Methyl 1-Benzamido-6-oxo-1,6-dihydropyridine-3-carboxylates: Assembly of the [1,2,4]Triazolo[1,5-a]pyridine Ring System

Published:2017-06-02 Issue:12 Volume:82 Page:6279-6288
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

Moloney Harold¹^ORCID,Magnus Nicholas A.¹,Buser Jonas Y.¹,Embry Matthew C.¹

Affiliation:

1. Small Molecule Design and Development, Eli Lilly and Company, Indianapolis, Indiana 46285, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.joc.7b00873

Reference37 articles.

1. Triazolopyridines as Selective JAK1 Inhibitors: From Hit Identification to GLPG0634

2. 2-Amino-[1,2,4]triazolo[1,5-a]pyridines as JAK2 inhibitors

3. A selective inhibitor reveals PI3Kγ dependence of TH17 cell differentiation

4. SAR studies around a series of triazolopyridines as potent and selective PI3Kγ inhibitors

5. Discovery of 5-(2-amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-(tert-butyl)pyridine-3-sulfonamide (CZC24758), as a potent, orally bioavailable and selective inhibitor of PI3K for the treatment of inflammatory disease

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