Atropodiastereoselective 5N-Acylation of 1,5-Benzodiazepin-2-ones with (S)-2-Phenylpropanoyl and (S)-2-Phenylbutanoyl Chlorides-Reference-Cited by-同舟云学术

Atropodiastereoselective 5N-Acylation of 1,5-Benzodiazepin-2-ones with (S)-2-Phenylpropanoyl and (S)-2-Phenylbutanoyl Chlorides

Published:2022-10-12 Issue:22 Volume:87 Page:15289-15300
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

Funaki Kaoru¹,Tabata Hidetsugu¹^ORCID,Nakazato Yusuke¹,Takahashi Yuka¹,Tasaka Tomohiko²,Takahashi Hideyo³^ORCID,Natsugari Hideaki²⁴^ORCID,Oshitari Tetsuta¹^ORCID

Affiliation:

1. Faculty of Pharma Sciences, Teikyo University, 2-11-1 Kaga, Itabashi-ku, Tokyo 173-8605, Japan

2. Affinity Science Corporation, 1-11-1 Nishi-Gotanda, Shinagawa-ku, Tokyo 141-0031, Japan

3. Faculty of Pharmaceutical Sciences, Tokyo University of Science, 2641 Yamazaki, Noda, Chiba 278-8510, Japan

4. Faculty of Pharmaceutical Sciences, The University of Tokyo, 7-3-1 Hongo, Bunkyo-ku, Tokyo 113-0033, Japan

Funder

Pharmaceutical Society of Japan

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.joc.2c01853

Reference28 articles.

1. Stereogenic and conformational properties of medium-ring benzo-fused N-heterocycle atropisomers

2. Recent encounters with atropisomerism in drug discovery

3. Atropisomerism in medicinal chemistry: challenges and opportunities

4. Nonbiaryl and Heterobiaryl Atropisomers: Molecular Templates with Promise for Atropselective Chemical Transformations

5. Assessing Atropisomer Axial Chirality in Drug Discovery and Development

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