Lewis Acid-Catalyzed Diastereoselective Synthesis of Multisubstituted N-Acylaziridine-2-carboxamides from 2H-Azirines via Joullié–Ugi Three-Component Reaction-Reference-Cited by-同舟云学术

Lewis Acid-Catalyzed Diastereoselective Synthesis of Multisubstituted N-Acylaziridine-2-carboxamides from 2H-Azirines via Joullié–Ugi Three-Component Reaction

Published:2018-03-02 Issue:7 Volume:83 Page:3570-3581
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

Angyal Anikó¹²,Demjén András¹²,Wéber Edit³,Kovács Anita K.⁴,Wölfling János²,Puskás László G.¹,Kanizsai Iván¹^ORCID

Affiliation:

1. AVIDIN Ltd., Alsó kikötő sor 11/D, Szeged H-6726, Hungary

2. Department of Organic Chemistry, University of Szeged, Dóm tér 8, Szeged H-6720, Hungary

3. SZTE-MTA Lendület Foldamer Research Group, Institute of Pharmaceutical Analysis, University of Szeged, Somogyi u. 4, Szeged H-6720, Hungary

4. Department of Medical Chemistry, University of Szeged, Dóm tér 8, Szeged 6720, Hungary

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.joc.7b03189

Reference64 articles.

1. Heterocycles in Natural Product Synthesis

2. Synthetic Aziridines in Medicinal Chemistry: A Mini-Review

3. On the synthesis of (2S)-aziridine-2-carboxylic acid containing peptides

4. A Convenient One-Pot Conversion of N-Boc-β-Aminoalcohols into N-Boc-Aziridines

5. Site-Selective Conjugation of Thiols with Aziridine-2-Carboxylic Acid-Containing Peptides

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