Synthesis of 1-(tert-Butyl) 4-Methyl (1R,2S,4R)-2-Methylcyclohexane-1,4-dicarboxylate from Hagemann’s tert-Butyl Ester for an Improved Synthesis of BMS-986251
Author:
Affiliation:
1. Research and Early Development, Bristol Myers Squibb Company, Princeton, New Jersey 08543-4000, United States
2. Materials Science & Engineering, Bristol Myers Squibb, 1 Squibb Drive, New Brunswick, New Jersey 08903, United States
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.joc.0c01169
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1. Design, synthesis and in vitro evaluation of novel uni- and bivalent ligands for the cannabinoid receptor type 1 with variation of spacer length and structure
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3. Higher order iminodiacetic acid libraries for probing protein-protein interactions
4. Diprovocims: A New and Exceptionally Potent Class of Toll-like Receptor Agonists
5. Synthesis and biological evaluation of aminothiazoles against Histoplasma capsulatum and Cryptococcus neoformans
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