Synthesis and QSAR of Quinazoline Sulfonamides As Highly Potent Human Histamine H4 Receptor Inverse Agonists-Reference-Cited by-同舟云学术

Synthesis and QSAR of Quinazoline Sulfonamides As Highly Potent Human Histamine H4 Receptor Inverse Agonists

Published:2010-03-01 Issue:6 Volume:53 Page:2390-2400
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Smits Rogier A.¹,Adami Maristella²,Istyastono Enade P.³,Zuiderveld Obbe P.³,van Dam Cindy M. E.³,de Kanter Frans J. J.³,Jongejan Aldo³,Coruzzi Gabriella²,Leurs Rob³,de Esch Iwan J. P.³

Affiliation:

1. Griffin Discoveries BV, Department of Medicinal Chemistry, Room P-246, De Boelelaan 1083, 1081 HV, Amsterdam, The Netherlands

2. Department of Human Anatomy, Pharmacology and Forensic Medicine, Section of Pharmacology, University of Parma, via Volturno 39, 43100 Parma, Italy

3. Leiden/Amsterdam Center for Drug Research (LACDR), Division of Medicinal Chemistry, Department of Pharmacochemistry, Faculty of Exact Sciences, Vrije Universiteit Amsterdam, De Boelelaan 1083, 1081 HV Amsterdam, The Netherlands

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm901379s

Reference32 articles.

1. Molecular Cloning and Characterization of a Novel Type of Histamine Receptor Preferentially Expressed in Leukocytes

2. The role of histamine H1 and H4 receptors in allergic inflammation: the search for new antihistamines

3. A Potent and Selective Histamine H4 Receptor Antagonist with Anti-Inflammatory Properties

4. Cloning, Expression, and Pharmacological Characterization of a Novel Human Histamine Receptor

5. Molecular Cloning and Characterization of a New Human Histamine Receptor, HH4R

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