Selective Non-nucleoside Inhibitors of Human DNA Methyltransferases Active in Cancer Including in Cancer Stem Cells-Reference-Cited by-同舟云学术

Selective Non-nucleoside Inhibitors of Human DNA Methyltransferases Active in Cancer Including in Cancer Stem Cells

Published:2014-01-15 Issue:3 Volume:57 Page:701-713
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Valente Sergio¹,Liu Yiwei²,Schnekenburger Michael³,Zwergel Clemens¹⁴,Cosconati Sandro⁵,Gros Christina⁶,Tardugno Maria¹,Labella Donatella¹,Florean Cristina³,Minden Steven³,Hashimoto Hideharu²,Chang Yanqi²,Zhang Xing²,Kirsch Gilbert⁴,Novellino Ettore⁷,Arimondo Paola B.⁶,Miele Evelina⁸,Ferretti Elisabetta⁹,Gulino Alberto⁹,Diederich Marc³¹⁰,Cheng Xiaodong²,Mai Antonello¹

Affiliation:

1. Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza Università di Roma, P.le Aldo Moro 5, 00185 Roma, Italy

2. Department of Biochemistry, Emory University School of Medicine, 1510 Clifton Road, Atlanta, Georgia 30322, United States

3. Laboratoire de Biologie Moléculaire et Cellulaire du Cancer (LBMCC), Hôpital Kirchberg, 9, rue Edward Steichen, L-2540 Luxembourg

4. Laboratoire d’Ingénierie Moléculaire et Biochimie Pharmacologique, Université de Lorraine−Metz, 1 Boulevard Arago, 57070 Metz, France

5. DiSTABiF, Seconda Università di Napoli, Via G. Vivaldi 43, 81100 Caserta, Italy

6. USR3388 CNRS-Pierre Fabre ETaC, CRDPF, 3 Avenue H. Curien, 31035 Toulouse Cedex 01, France

7. Dipartimento di Farmacia, Università di Napoli “Federico II”, Via D. Montesano, 49, 80131 Napoli, Italy

8. Istituto Italiano di Tecnologia and Dipartimento of Medicina Molecolare, Sapienza Università di Roma, Viale Regina Elena 291, 00161 Roma, Italy

9. Dipartimento di Medicina Sperimentale e Dipartimento di Medicina Molecolare, Sapienza Università di Roma, Viale Regina Elena 291, 00161 Rome, Italy

10. Department of Pharmacy, College of Pharmacy, Seoul National University, 599 Gwanak-ro, Gwanak-gu, Seoul 151-742, Korea

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm4012627

Reference44 articles.

1. Epigenetic protein families: a new frontier for drug discovery

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5. Epigenomics of leukemia: from mechanisms to therapeutic applications

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