Implementation of a High-Temperature Claisen Approach for Early Phase Delivery of a Benzopyran Derivative-Reference-Cited by-同舟云学术

Implementation of a High-Temperature Claisen Approach for Early Phase Delivery of a Benzopyran Derivative

Published:2009-12-07 Issue:1 Volume:14 Page:85-91
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Walker Andrew J.¹,Adolph Sven¹,Connell Richard B.¹,Laue Klaus¹,Roeder Michael¹,Rueggeberg Carsten J.¹,Hahn Dirk Uwe¹,Voegtli Kurt¹,Watson John¹

Affiliation:

1. Carbogen-AMCIS AG, Neulandweg 5, CH-5502, Hunzenschwil, Switzerland, GlaxoSmithKline Medicines Research Centre, Gunnels Wood Road, Stevenage, Herfordshire SG1 2NY, United Kingdom, Carbogen-AMCIS AG, Hauptstrasse 171, CH-4416, Bubendorf, Switzerland, and Carbogen-AMCIS AG, Schachenallee 29, CH-5001, Aarau, Switzerland

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/op900193v

Reference15 articles.

1. aAhmed, M., Miller, N. D., Moss, S. F., and Sanger, G. J.WO 2007096352, 2007.

2. 5-HT4 receptor agonists: similar but not the same

3. cFor tegaserod, see:

4. Experimental pancreatitis disturbs gastrointestinal and colonic motility in mice: effect of the prokinetic agent tegaserod

5. Investigation of Synthetic Routes to a Key Benzopyran Intermediate of a 5HT4 Agonist

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