A Novel, High-Affinity, Fluorescent Progesterone Receptor Antagonist. Synthesis and in Vitro Studies-Reference-Cited by-同舟云学术

A Novel, High-Affinity, Fluorescent Progesterone Receptor Antagonist. Synthesis and in Vitro Studies

Published:2004-02-26 Issue:2 Volume:15 Page:359-365
ISSN:1043-1802
Container-title:Bioconjugate Chemistry
language:en
Short-container-title:Bioconjugate Chem.

Author:

Hödl Claudia¹,Strauss Wolfgang S. L.¹,Sailer Reinhard¹,Seger Christoph¹,Steiner Rudolf¹,Haslinger Ernst¹,Schramm H. Wolfgang¹

Affiliation:

1. Institute for Pharmaceutical Chemistry and Pharmaceutical Technology, Karl-Franzens-University, Universitätsplatz 1, A-8010 Graz, Austria, Institut für Lasertechnologien in der Medizin und Messtechnik an der Universität Ulm, Helmholtzstrasse 12, D-89081 Ulm, Germany, and Institute of Pharmacy, Department of Pharmacognosy, Leopold-Franzens-University, Innrain 52, A-6020 Innsbruck, Austria

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Pharmaceutical Science,Pharmacology,Biomedical Engineering,Bioengineering,Biotechnology

Link

https://pubs.acs.org/doi/pdf/10.1021/bc034169o

Reference45 articles.

1. Investigation of the binding interactions of progesterone using muteins of the human progesterone receptor ligand binding domain designed on the basis of a three-dimensional protein model

2. Synthesis and Biological Activity of a Novel, Highly Potent Progesterone Receptor Antagonist

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