Isocombretastatins A versus Combretastatins A: The Forgotten isoCA-4 Isomer as a Highly Promising Cytotoxic and Antitubulin Agent-Reference-Cited by-同舟云学术

Isocombretastatins A versus Combretastatins A: The Forgotten isoCA-4 Isomer as a Highly Promising Cytotoxic and Antitubulin Agent

Published:2009-06-16 Issue:14 Volume:52 Page:4538-4542
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Messaoudi Samir¹,Tréguier Bret¹,Hamze Abdallah¹,Provot Olivier¹,Peyrat Jean-François¹,De Losada Jordi Rodrigo¹,Liu Jian-Miao²,Bignon Jérôme²,Wdzieczak-Bakala Joanna²,Thoret Sylviane²,Dubois Joëlle²,Brion Jean-Daniel¹,Alami Mouâd¹

Affiliation:

1. Univ Paris-Sud, CNRS, BioCIS-UMR 8076, Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie, 5 rue J.-B. Clément, Châtenay-Malabry F-92296, France

2. Institut de Chimie des Substances Naturelles (ICSN), UPR 2301 CNRS, Avenue de la Terrasse, F-91198 Gif-sur-Yvette, France

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm900321u

Reference26 articles.

1. Alami, M.; Brion, J.D.; Provot, O.; Peyrat, J.F.; Messaoudi, S.; Hamze, A.; Giraud, A.; Bignon, J.; Bakala, J.; Liu, J.M.IsoCA-4 and analogues thereof as potent cytotoxic agents inhibiting tubulin polymerization. Patent WO 122620 A1, 2008.

2. Promotion of microtubule assembly in vitro by taxol

3. Anti-mitotic activity of colchicine and the structural basis for its interaction with tubulin

4. Current Status of Oral Carbapenem Development

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