Synthesis, Structure−Activity Relationship, and Receptor Pharmacology of a New Series of Quinoline Derivatives Acting as Selective, Noncompetitive mGlu1 Antagonists-Reference-Cited by-同舟云学术

Synthesis, Structure−Activity Relationship, and Receptor Pharmacology of a New Series of Quinoline Derivatives Acting as Selective, Noncompetitive mGlu1 Antagonists

Published:2005-01-28 Issue:6 Volume:48 Page:2134-2153
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Mabire Dominique¹,Coupa Sophie¹,Adelinet Christophe¹,Poncelet Alain¹,Simonnet Yvan¹,Venet Marc¹,Wouters Ria¹,Lesage Anne S. J.¹,Beijsterveldt Ludy Van¹,Bischoff François¹

Affiliation:

1. Department of Medicinal Chemistry, Johnson & Johnson Pharmaceutical Research & Development, a Division of Janssen-Cilag France, Campus de Maigremont, F-27106 Val de Reuil, France, and Department of Medicinal Chemistry, CNS Discovery Research and Department of Preclinical Pharmacokinetics, Johnson & Johnson Pharmaceutical Research & Development, a Division of Janssen Pharmaceutica N.V., Turnhoutseweg 30, B-2340 Beerse, Belgium

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm049499o

Reference48 articles.

1. Distribution of metabotropic glutamate receptor mGluR5 immunoreactivity in rat brain

2. Cloned Glutamate Receptors

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