Mimicking the Intramolecular Hydrogen Bond: Synthesis, Biological Evaluation, and Molecular Modeling of Benzoxazines and Quinazolines as Potential Antimalarial Agents-Reference-Cited by-同舟云学术

Mimicking the Intramolecular Hydrogen Bond: Synthesis, Biological Evaluation, and Molecular Modeling of Benzoxazines and Quinazolines as Potential Antimalarial Agents

Published:2012-11-21 Issue:23 Volume:55 Page:10387-10404
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Gemma Sandra¹²,Camodeca Caterina¹²,Brindisi Margherita¹²,Brogi Simone¹²,Kukreja Gagan¹²,Kunjir Sanil¹²,Gabellieri Emanuele¹²,Lucantoni Leonardo²³,Habluetzel Annette²³,Taramelli Donatella¹²,Basilico Nicoletta¹²,Gualdani Roberta⁴,Tadini-Buoninsegni Francesco⁴,Bartolommei Gianluca⁴,Moncelli Maria Rosa⁴,Martin Rowena E.⁵,Summers Robert L.⁵,Lamponi Stefania¹²,Savini Luisa¹²,Fiorini Isabella¹²,Valoti Massimo⁶,Novellino Ettore¹⁷,Campiani Giuseppe¹²,Butini Stefania¹²

Affiliation:

1. European Research Centre for Drug Discovery and Development (NatSynDrugs), University of Siena, Via Aldo Moro, 53100 Siena, Italy

2. CIRM Centro Interuniversitario di Ricerche sulla Malaria, Università di Torino, Torino, Italy

3. Scuola di Scienze del Farmaco e dei Prodotti della Salute, Università di Camerino, 62032 Camerino (MC), Italy

4. Department of Chemistry “Ugo Schiff”, University of Florence, 50019 Sesto Fiorentino, Italy

5. Research School of Biology, The Australian National University, Canberra ACT 0200, Australia

6. Dipartimento di Neuroscienze, University of Siena, via A. Moro 2, Siena, Italy

7. Dipartimento di Chimica Farmaceutica e Tossicologica, University of Naples Federico II, Via D. Montesano 49, 80131 Naples, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm300831b

Reference83 articles.

1. WHO World Malaria Report 2011;World Health Organization:Geneva, 2011; http://www.who.int/malaria/world_malaria_report_2011/en/.

2. Global malaria mortality between 1980 and 2010: a systematic analysis

3. EFFECTIVENESS OF AMODIAQUINE AS TREATMENT FOR CHLOROQUINE-RESISTANT PLASMODIUM FALCIPARUM INFECTIONS IN KENYA

4. Systematic review of amodiaquine treatment in uncomplicated malaria

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