Identification of a 4-(Hydroxymethyl)diarylhydantoin as a Selective Androgen Receptor Modulator-Reference-Cited by-同舟云学术

Identification of a 4-(Hydroxymethyl)diarylhydantoin as a Selective Androgen Receptor Modulator

Published:2012-09-25 Issue:19 Volume:55 Page:8236-8247
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Nique François¹,Hebbe Séverine¹,Triballeau Nicolas¹,Peixoto Christophe¹,Lefrançois Jean-Michel¹,Jary Hélène¹,Alvey Luke¹,Manioc Murielle¹,Housseman Christopher¹,Klaassen Hugo¹,Van Beeck Kris¹,Guédin Denis¹,Namour Florence¹,Minet Dominque¹,Van der Aar Ellen¹,Feyen Jean¹,Fletcher Stephen¹,Blanqué Roland¹,Robin-Jagerschmidt Catherine¹,Deprez Pierre¹

Affiliation:

1. GALAPAGOS, Parc Biocitech, 102 Avenue Gaston Roussel, 93230 Romainville, France

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm300281x

Reference31 articles.

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2. bBrueggemier, R. W.; Miller, D. D.; Witiak, D. T.InPrinciples of Medicinal Chemistry, 4th ed.Foye, W. O.; Lemke, T. L.; Williams, D. A., Eds.Williams and Wilkins:Baltimore, MD, 1995; Chapter 23, pp486–493.

3. Risks Versus Benefits of Testosterone Therapy in Elderly Men

4. Risks of Testosterone-Replacement Therapy and Recommendations for Monitoring

5. Testosterone and Prostate Cancer: An Historical Perspective on a Modern Myth

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