Galactosyl Prodrug of Ketorolac: Synthesis, Stability, and Pharmacological and Pharmacokinetic Evaluations-Reference-Cited by-同舟云学术

Galactosyl Prodrug of Ketorolac: Synthesis, Stability, and Pharmacological and Pharmacokinetic Evaluations

Published:2009-05-21 Issue:12 Volume:52 Page:3794-3800
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Curcio Annalisa¹,Sasso Oscar¹,Melisi Daniela¹,Nieddu Maria¹,La Rana Giovanna¹,Russo Roberto¹,Gavini Elisabetta¹,Boatto Gianpiero¹,Abignente Enrico¹,Calignano Antonio¹,Rimoli Maria Grazia¹

Affiliation:

1. Department of Pharmaceutical and Toxicological Chemistry and Department of Experimental Pharmacology, Faculty of Pharmacy, Federico II University of Naples, Via Domenico Montesano 49, 80131, Naples, Italy, and Department of Drug, Chemistry and Toxicology and Department of Drug Sciences, Faculty of Pharmacy, University of Sassari, Via Muroni 23/a, 07100, Sassari, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm900051r

Reference27 articles.

1. Ketorolac

2. Upper Gastrointestinal Bleeding Associated with the Use of NSAIDs

3. A prospective study comparing i.m. ketorolac with i.m. meperidine in the treatment of acute biliary colic

4. The role of direct tissue contact in the production of gastrointestinal ulcers by anti-inflammatory drugs in rats

5. Mechanisms of Gastrointestinal Toxicity of Nonsteroidal Anti-Inflammatory Drugs

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