A Backbone-Cyclic, Receptor 5-Selective Somatostatin Analogue: Synthesis, Bioactivity, and Nuclear Magnetic Resonance Conformational Analysis-Reference-Cited by-同舟云学术

A Backbone-Cyclic, Receptor 5-Selective Somatostatin Analogue: Synthesis, Bioactivity, and Nuclear Magnetic Resonance Conformational Analysis

Published:1998-02-24 Issue:6 Volume:41 Page:919-929
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Gilon Chaim¹,Huenges Martin¹,Mathä Barbara¹,Gellerman Gary¹,Hornik Vered¹,Afargan Michel¹,Amitay Oved¹,Ziv Ofer¹,Feller Etty¹,Gamliel Asher¹,Shohat Dvira¹,Wanger Mazal¹,Arad Oded¹,Kessler Horst¹

Affiliation:

1. Department of Organic Chemistry, Hebrew University, Jerusalem, Israel, Institut für Organische Chemie und Biochemie, Technische Universität München, Lichtenbergstrasse 4, D-85747 Garching, Germany, and Peptor Ltd., Kiryat Weizmann, Rehovot 76326, Israel

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm970633x

Reference25 articles.

1. Backbone cyclization: A new method for conferring conformational constraint on peptides

2. New backbone cyclic substance P analogs

3. Stereocontrolled synthesis of C2-symmetric and pseudo-C2-symmetric diamino alcohols and diols for use in HIV protease inhibitors

4. Conformation of cyclic analogs of substance P: NMR and molecular dynamics in dimethyl sulfoxide

5. Comparison of the Conformation of Active and Nonactive Backbone Cyclic Analogs of Substance P as a Tool To Elucidate Features of the Bioactive Conformation: NMR and Molecular Dynamics in DMSO and Water

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