Diastereoselective Synthesis of New ψ[(E)-CHCMe]- and ψ[(Z)-CHCMe]-type Alkene Dipeptide Isosteres by Organocopper Reagents and Application to Conformationally Restricted Cyclic RGD Peptidomimetics-Reference-Cited by-同舟云学术

Diastereoselective Synthesis of New ψ[(E)-CHCMe]- and ψ[(Z)-CHCMe]-type Alkene Dipeptide Isosteres by Organocopper Reagents and Application to Conformationally Restricted Cyclic RGD Peptidomimetics

Published:2002-08-01 Issue:17 Volume:67 Page:6162-6173
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

Oishi Shinya¹,Kamano Takae¹,Niida Ayumu¹,Odagaki Yoshihiko¹,Hamanaka Nobuyuki¹,Yamamoto Mikio¹,Ajito Keiichi¹,Tamamura Hirokazu¹,Otaka Akira¹,Fujii Nobutaka¹

Affiliation:

1. Graduate School of Pharmaceutical Sciences, Kyoto University, Sakyo-ku, Kyoto, 606-8501, Japan, Minase Research Institute, Ono Pharmaceutical Co. Ltd., Mishima-gun, Osaka, 618-8585, Japan, and Pharmaceutical Research Center, Meiji Seika Kaisha, Ltd., Kohoku-ku, Yokohama, 222-0002, Japan

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/jo025923m

Reference74 articles.

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2. Integrin Structure

3. Requirement of Vascular Integrin α v β 3 for Angiogenesis

4. Integrins and cancer

5. Interactions between the bone matrix proteins osteopontin and bone sialoprotein and the osteoclast integrin alpha v beta 3 potentiate bone resorption

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