Metabolism-Based Identification of a Potent Thrombin Receptor Antagonist-Reference-Cited by-同舟云学术

Metabolism-Based Identification of a Potent Thrombin Receptor Antagonist

Published:2006-12-13 Issue:1 Volume:50 Page:129-138
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Clasby Martin C.¹,Chackalamannil Samuel¹,Czarniecki Michael¹,Doller Dario¹,Eagen Keith¹,Greenlee William¹,Kao Grace¹,Lin Yan¹,Tsai Hsingan¹,Xia Yan¹,Ahn Ho-Sam¹,Agans-Fantuzzi Jacqueline¹,Boykow George¹,Chintala Madhu¹,Foster Carolyn¹,Smith-Torhan April¹,Alton Kevin¹,Bryant Matthew¹,Hsieh Yunsheng¹,Lau Janice¹,Palamanda Jairam¹

Affiliation:

1. Central Nervous System and Cardiovascular Chemical Research, Cardiovascular and Metabolic Disease Research, and Drug Metabolism and Pharmacokinetics Research, Schering-Plough Research Institute, 2015 Galloping Hill Road, Kenilworth, New Jersey 07033

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm061043e

Reference31 articles.

1. The coagulation cascade: initiation, maintenance, and regulation

2. Cellular effects of thrombin: pharmacology of the receptor(s) in various cell types and possible development of receptor antagonists

3. Thrombin-Cellular Interactions

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