Design, Synthesis, and Biological Evaluation of Novel Investigational Nonapeptide KISS1R Agonists with Testosterone-Suppressive Activity-Reference-Cited by-同舟云学术

Design, Synthesis, and Biological Evaluation of Novel Investigational Nonapeptide KISS1R Agonists with Testosterone-Suppressive Activity

Published:2013-10-17 Issue:21 Volume:56 Page:8298-8307
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Asami Taiji¹,Nishizawa Naoki¹,Matsui Hisanori¹,Nishibori Kimiko¹,Ishibashi Yoshihiro¹,Horikoshi Yasuko¹,Nakayama Masaharu¹,Matsumoto Shin-ichi¹,Tarui Naoki¹,Yamaguchi Masashi¹,Matsumoto Hirokazu¹,Ohtaki Tetsuya¹,Kitada Chieko¹

Affiliation:

1. Pharmaceutical Research Division, Shonan Research Center, Takeda Pharmaceutical Company Ltd, 2-26-1, Muraoka-Higashi Fujisawa, Kanagawa 251-8555, Japan

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm401056w

Reference17 articles.

1. Metastasis suppressor gene KiSS-1 encodes peptide ligand of a G-protein-coupled receptor

2. The Metastasis Suppressor Gene KiSS-1 Encodes Kisspeptins, the Natural Ligands of the Orphan G Protein-coupled Receptor GPR54

3. AXOR12, a Novel Human G Protein-coupled Receptor, Activated by the Peptide KiSS-1

4. Discovery of a receptor related to the galanin receptors

5. Peripheral administration of metastin induces marked gonadotropin release and ovulation in the rat

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