Novel Potent and Selective Central 5-HT3 Receptor Ligands Provided with Different Intrinsic Efficacy. 2. Molecular Basis of the Intrinsic Efficacy of Arylpiperazine Derivatives at the Central 5-HT3 Receptors-Reference-Cited by-同舟云学术

Novel Potent and Selective Central 5-HT3 Receptor Ligands Provided with Different Intrinsic Efficacy. 2. Molecular Basis of the Intrinsic Efficacy of Arylpiperazine Derivatives at the Central 5-HT3 Receptors

Published:1999-04-10 Issue:9 Volume:42 Page:1556-1575
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Cappelli Andrea¹,Anzini Maurizio¹,Vomero Salvatore¹,Canullo Laura¹,Mennuni Laura¹,Makovec Francesco¹,Doucet Edith¹,Hamon Michel¹,Menziani M. Cristina¹,De Benedetti Pier G.¹,Bruni Giancarlo¹,Romeo Maria R.¹,Giorgi Gianluca¹,Donati Alessandro¹

Affiliation:

1. Dipartimento Farmaco Chimico Tecnologico, Università di Siena, Via Banchi di Sotto 55, 53100 Siena, Italy, Facoltà di Farmacia, Università degli Studi di Catanzaro “Magna Graecia”, Complesso Ninì Barbieri, 88021 Roccelletta di Borgia, Catanzaro, Italy, Rotta Research Laboratorium S.p.A., Via Valosa di Sopra 7, 20052 Monza, Italy, Neurobiologie Cellulaire et Fonctionnelle, INSERM U. 288, Faculté de Médicine Pitié-Salpêtriére, 91, Boulevard de l'Hôpital, 75634 Paris Cedex 13, France, Dipartimento di...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm981112s

Reference54 articles.

1. 5-HT3 receptors

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4. Cholecystokinin release mediated by 5-HT3 receptors in rat cerebral cortex and nucleus accumbens

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