Peptido Sulfonyl Fluorides as New Powerful Proteasome Inhibitors-Reference-Cited by-同舟云学术

Peptido Sulfonyl Fluorides as New Powerful Proteasome Inhibitors

Published:2012-12-13 Issue:24 Volume:55 Page:10995-11003
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Brouwer Arwin J.¹,Jonker Anika¹,Werkhoven Paul¹,Kuo Ethan²,Li Nan²,Gallastegui Nerea³,Kemmink Johan¹,Florea Bogdan I.²,Groll Michael³,Overkleeft Herman S.²,Liskamp Rob M. J.¹

Affiliation:

1. Department of Medicinal Chemistry and Chemical Biology, Utrecht Institute for Pharmaceutical Sciences, Faculty of Science, Utrecht University, P.O. Box 80082, 3508 TB Utrecht, The Netherlands

2. Bio-organic synthesis, Leiden Institute of Chemistry, Leiden University, P.O. Box 9502, 2300 RA, Leiden, The Netherlands

3. Center for Integrated Protein Science at the Department Chemie, Lehrstuhl für Biochemie, Technische Universität München, Lichtenbergstrasse 4, 85748, Garching, Germany.

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm301443r

Reference22 articles.

1. Contribution of Proteasomal β-Subunits to the Cleavage of Peptide Substrates Analyzed with Yeast Mutants

2. Potent and selective inhibitors of the proteasome: Dipeptidyl boronic acids

3. Development of the Proteasome Inhibitor Velcade™ (Bortezomib)

4. Novel Proteasome Inhibitors to Overcome Bortezomib Resistance

5. Opening the door to a new class of proteasome inhibitors

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