“True” Antiandrogens—Selective Non-Ligand-Binding Pocket Disruptors of Androgen Receptor–Coactivator Interactions: Novel Tools for Prostate Cancer-Reference-Cited by-同舟云学术

“True” Antiandrogens—Selective Non-Ligand-Binding Pocket Disruptors of Androgen Receptor–Coactivator Interactions: Novel Tools for Prostate Cancer

Published:2012-02-10 Issue:4 Volume:55 Page:1635-1644
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Caboni Laura¹,Kinsella Gemma K.¹,Blanco Fernando¹,Fayne Darren¹,Jagoe William N.¹,Carr Miriam¹,Williams D. Clive¹,Meegan Mary J.¹,Lloyd David G.¹

Affiliation:

1. Molecular Design Group, School of Biochemistry and Immunology, ‡School of Biochemistry and Immunology, and §School of Pharmacy and Pharmaceutical Sciences, Trinity Biomedical Sciences Institute, Trinity College Dublin, Dublin 2, Ireland

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm201438f

Reference52 articles.

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3. Nuclear Receptor Structure: Implications for Function

4. A surface on the androgen receptor that allosterically regulates coactivator binding

5. Anti-androgens and androgen-depleting therapies in prostate cancer: new agents for an established target

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