Iridals Are a Novel Class of Ligands for Phorbol Ester Receptors with Modest Selectivity for the RasGRP Receptor Subfamily

Author:

Shao Lei1,Lewin Nancy E.1,Lorenzo Patricia S.1,Hu Zengjian1,Enyedy Istvan J.1,Garfield Susan H.1,Stone James C.1,Marner Franz-Josef1,Blumberg Peter M.1,Wang Shaomeng1

Affiliation:

1. Drug Discovery Program, University of Michigan Cancer Center, Departments of Internal Medicine and Medicinal Chemistry, University of Michigan, 1500 E. Medical Center Drive, Ann Arbor, Michigan 48109-0934, Laboratory of Cellular Carcinogenesis and Tumor Promotion and Laboratory of Experimental Carcinogenesis, National Cancer Institute, Bethesda, Maryland 20892, Institute of Biochemistry, University of Cologne, Cologne, Germany D-50674, and Department of Biochemistry, University of Alberta, Edmonton,...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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