Discovery of the Selective CYP17A1 Lyase Inhibitor BMS-351 for the Treatment of Prostate Cancer-Reference-Cited by-同舟云学术

Discovery of the Selective CYP17A1 Lyase Inhibitor BMS-351 for the Treatment of Prostate Cancer

Published:2015-12-14 Issue:1 Volume:7 Page:40-45
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Huang Audris¹,Jayaraman Lata¹,Fura Aberra¹,Vite Gregory D.¹,Trainor George L.¹,Gottardis Marco M.¹,Spires Thomas E.¹,Spires Vanessa M.¹,Rizzo Cheryl A.¹,Obermeier Mary T.¹,Elzinga Paul A.¹,Todderud Gordon¹,Fan Yi¹,Newitt John A.¹,Beyer Sophie M.¹,Zhu Yongxin¹,Warrack Bethanne M.¹,Goodenough Angela K.¹,Tebben Andrew J.¹,Doweyko Arthur M.¹,Gold David L.¹,Balog Aaron¹

Affiliation:

1. Bristol-Myers Squibb Research and Development, Princeton, New Jersey 08543-4000, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.5b00310

Reference21 articles.

1. National Cancer Institute website. Cancer Topics: Prostate Cancer.http://www.cancer.gov/cancertopics/types/prostate(accessed 2015, May 28).

2. EFFECT OF ORCHIECTOMY AND IRRADIATION ON CANCER OF THE PROSTATE

3. Targeting the Adrenal Gland in Castration-Resistant Prostate Cancer: A Case for Orteronel, a Selective CYP-17 17,20-Lyase Inhibitor

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