Affinity-Based Fluorescence Polarization Assay for High-Throughput Screening of Prolyl Hydroxylase 2 Inhibitors-Reference-Cited by-同舟云学术

Affinity-Based Fluorescence Polarization Assay for High-Throughput Screening of Prolyl Hydroxylase 2 Inhibitors

Published:2015-11-12 Issue:12 Volume:6 Page:1236-1240
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Lei Yonghua¹,Hu Tianhan¹,Wu Xingsen¹,Wu Yue¹,Bao Qichao¹,Zhang Lianshan²,Xia Hua¹,Sun Haopeng¹,You Qidong¹,Zhang Xiaojin¹³

Affiliation:

1. Jiangsu Key Laboratory of Drug Design and Optimization, and State Key Laboratory of Natural Medicines, China Pharmaceutical University, Nanjing 210009, China

2. National Engineering and Research Center for Target Drugs, Lianyungang 222000, China

3. Department of Organic Chemistry, School of Science, China Pharmaceutical University, Nanjing 210009, China

Funder

Priority Academic Program Development of Jiangsu Higher Education Institutions

National Natural Science Foundation of China

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.5b00394

Reference27 articles.

1. Structure-based drug design for hypoxia-inducible factor prolyl-hydroxylase inhibitors and its therapeutic potential for the treatment of erythropoiesis-stimulating agent-resistant anemia: raising expectations for exploratory clinical trials

2. HIF prolyl hydroxylase inhibitors for anemia

3. The human oxygen sensing machinery and its manipulation

4. Oxygen Sensing by Metazoans: The Central Role of the HIF Hydroxylase Pathway

5. Oxygen sensing by HIF hydroxylases

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