Discovery and Optimization of Seven-Membered Lactam-Based Compounds to Phenocopy the Inhibition of the Aurora Kinase B-Reference-Cited by-同舟云学术

Discovery and Optimization of Seven-Membered Lactam-Based Compounds to Phenocopy the Inhibition of the Aurora Kinase B

Published:2022-06-06 Issue:7 Volume:13 Page:1091-1098
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Huang Jian¹,Shi Qiong¹,Choudhry Namrta¹,Li Hongmei¹,Yang Chenglu¹,Kalashova Julia¹,Yan Ziqi¹,Li Jinhua¹,Reddy Mallu Chenna²,Gopala Sridhar Goud²,Zhang Shenqiu³,Zhang Jing¹,Nimishetti Naganna¹,Yang Dun¹^ORCID

Affiliation:

1. Chengdu Anticancer Bioscience, J. Michael Bishop Institute of Cancer Research, Chengdu, Sichuan 610000, China

2. Anticancer Bioscience (India), Hyderabad, Telangana 500051, India

3. Anticancer Bioscience (U.K.), St Andrews KY16 9QD, United Kingdom

Funder

Anticancer Bioscience

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.2c00098

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