Lipase-Catalyzed Synthesis and Biological Evaluation of N-Picolineamides as Trypanosoma cruzi Antiproliferative Agents

Author:

García Fabricio Freije1ORCID,Musikant Daniel2,Escalona José L.2,Edreira Martín M.2,Liñares Guadalupe García1ORCID

Affiliation:

1. Laboratorio de Biocatálisis, Departamento de Química Orgánica y UMYMFOR, Facultad de Ciencias Exactas y Naturales, Universidad de Buenos Aires-CONICET, Ciudad Universitaria, Pabellón 2, piso 3, C1428EGA Buenos Aires, Argentina

2. Laboratorio de Biología Molecular de Trypanosomas, Departamento de Química Biológica e IQUIBICEN, Facultad de Ciencias Exactas y Naturales, Universidad de Buenos Aires-CONICET, Ciudad Universitaria, Pabellón 2, piso 4, C1428EGA Buenos Aires, Argentina

Funder

Consejo Nacional de Investigaciones Cient?ficas y T?cnicas

Universidad de Buenos Aires

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Reference57 articles.

1. Specific chemotherapy of Chagas disease: Relevance, current limitations and new approaches

2. Organization, W. H. Fourth WHO report on neglected tropical diseases; WHO, 2017.

3. Organization, W. H. Chagas disease (also known as American trypanosomiasis). Online at https://www.who.int/news-room/fact-sheets/detail/chagas-disease-(american-trypanosomiasis) (accessed 2022-06-09).

4. Progresses in the Field of Drug Design to Combat Tropical Protozoan Parasitic Diseases

5. Other forms of transmission

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