Ligand Screening System for the RXRα Heterodimer Using the Fluorescence RXR Agonist CU-6PMN-Reference-Cited by-同舟云学术

Ligand Screening System for the RXRα Heterodimer Using the Fluorescence RXR Agonist CU-6PMN

Published:2023-02-20 Issue:3 Volume:14 Page:291-296
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Kawasaki Mayu¹,Motoyama Tomoharu¹,Yamada Shoya²,Watanabe Masaki²,Fujihara Michiko²,Kambe Akira¹,Nakano Shogo¹³^ORCID,Kakuta Hiroki²^ORCID,Ito Sohei¹

Affiliation:

1. Graduate School of Integrated Pharmaceutical and Nutritional Sciences, University of Shizuoka, 52-1 Yada, Suruga-ku, Shizuoka 422-8526, Japan

2. Division of Pharmaceutical Sciences, Okayama University Graduate School of Medicine, Dentistry and Pharmaceutical Sciences, 1-1-1, Tsushima-naka, Kita-ku, Okayama 700-8530, Japan

3. PREST, Japan Science and Technology Agency, Saitama 332-0012, Japan

Funder

Precursory Research for Embryonic Science and Technology

Japan Society for the Promotion of Science

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.2c00509

Reference30 articles.

1. Nuclear Receptors, RXR, and the Big Bang

2. Structural Overview of the Nuclear Receptor Superfamily: Insights into Physiology and Therapeutics

3. RXR alpha mutant mice establish a genetic basis for vitamin A signaling in heart morphogenesis.

4. Bexarotene Is Effective and Safe for Treatment of Refractory Advanced-Stage Cutaneous T-Cell Lymphoma: Multinational Phase II-III Trial Results

5. Development of Scaled-Up Synthetic Method for Retinoid X Receptor Agonist NEt-3IB Contributing to Sustainable Development Goals

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