Design, Synthesis, and Antitumor Evaluation of 4-Amino-(1H)-pyrazole Derivatives as JAKs Inhibitors-Reference-Cited by-同舟云学术

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Design, Synthesis, and Antitumor Evaluation of 4-Amino-(1H)-pyrazole Derivatives as JAKs Inhibitors

Published:2016-08-24 Issue:10 Volume:7 Page:950-955
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Liang Xuewu¹,Zang Jie¹,Zhu Mengyuan²,Gao Qianwen¹,Wang Binghe²,Xu Wenfang¹,Zhang Yingjie¹

Affiliation:

1. Department of Medicinal Chemistry, School of Pharmacy, Shandong University, Ji’nan, Shandong 250012, P. R. China

2. Department of Chemistry and Center for Diagnostics and Therapeutics, Georgia State University, Atlanta, Georgia 30303, United States

Funder

Ministry of Science and Technology of the People's Republic of China

Shandong Province

China Postdoctoral Science Foundation

Shandong University

National Natural Science Foundation of China

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.6b00247

Reference22 articles.

1. Discovery and Development of Janus Kinase (JAK) Inhibitors for Inflammatory Diseases

2. Defects in Jak-STAT-mediated cytokine signals cause hyper-IgE syndrome: lessons from a primary immunodeficiency

3. AT9283, a potent inhibitor of the Aurora kinases and Jak2, has therapeutic potential in myeloproliferative disorders

4. New and Old Functions of STAT3: A Pivitol Target for Individualized Treatment of Cancer

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1. A Review on Pyrazole Derivatives Used in the Treatment of Rheumatoid Arthritis: Recent Advancement and Drug Development;Current Rheumatology Reviews;2024-03-05

2. Targeting JAK2/STAT3 for the treatment of cancer: A review on recent advancements in molecular development using structural analysis and SAR investigations;Bioorganic Chemistry;2024-02

3. Exploration of Janus Kinase (JAK) and Histone Deacetylase (HDAC) Bispecific Inhibitors Based on the Moiety of Fedratinib for Treatment of Both Hematologic Malignancies and Solid Cancers;Journal of Medicinal Chemistry;2023-04-14

4. Pharmacophore-Based Virtual Screening and Experimental Validation of Pyrazolone-Derived Inhibitors toward Janus Kinases;ACS Omega;2022-09-06

5. Dual-target Janus kinase (JAK) inhibitors: Comprehensive review on the JAK-based strategies for treating solid or hematological malignancies and immune-related diseases;European Journal of Medicinal Chemistry;2022-09

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