From Dynamic Combinatorial Chemistry to in Vivo Evaluation of Reversible and Irreversible Myeloperoxidase Inhibitors

Author:

Soubhye Jalal1,Gelbcke Michel1,Van Antwerpen Pierre1,Dufrasne François1,Boufadi Mokhtaria Yasmina12,Nève Jean1,Furtmüller Paul G.3,Obinger Christian3,Zouaoui Boudjeltia Karim4,Meyer Franck5ORCID

Affiliation:

1. Chimie Pharmaceutique Organique, Faculty of pharmacy, Université Libre de Bruxelles (ULB), Boulevard du Triomphe, 1050 Bruxelles, Belgium

2. Laboratory of Beneficial Microorganisms, Functional Food and Health (LMBAFS), Faculty of Natural Sciences and Life, Université de Abdelhamid Ibn Badis, 27000 Mostaganem, Algeria

3. Department of Chemistry, BOKU−University of Natural Resources and Life Sciences, 1190 Vienna, Austria

4. Laboratory of Experimental Medicine (ULB 222 unit), Université Libre de Bruxelles, Chu de Charleroi, 6110 Belgium

5. Laboratory of Biopolymers and Supramolecular Nanomaterials, Faculty of Pharmacy, Université Libre de Bruxelles (ULB), Boulevard du Triomphe, 1050 Bruxelles, Belgium

Funder

Fonds De La Recherche Scientifique - FNRS

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

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