2-Trifluoromethylthiazole-5-carboxamides: Analogues of a Stilbene-Based Anti-HIV Agent that Impact HIV mRNA Processing-Reference-Cited by-同舟云学术

2-Trifluoromethylthiazole-5-carboxamides: Analogues of a Stilbene-Based Anti-HIV Agent that Impact HIV mRNA Processing

Published:2021-10-29 Issue:11 Volume:12 Page:1818-1823
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Zamiri Maryam¹,Cheung Peter K.²³,Brockman Mark A.²³,Brumme Zabrina L.²³,Chabot Benoit⁴,Cochrane Alan⁵,Grierson David S.¹^ORCID

Affiliation:

1. Faculty of Pharmaceutical Sciences, University of British Columbia, Vancouver, BC V6T 1Z3, Canada

2. BC Centre for Excellence in HIV/AIDS, 608−1081 Burrard Street, Vancouver, BC V6Z 1Y6, Canada

3. Faculty of Health Sciences, Simon Fraser University, Burnaby, BC V5A 1S6, Canada

4. Department of Microbiology and Infectious Diseases, Faculty of Medicine and Health Sciences, Université de Sherbrooke, Sherbrooke, QC J1E 4K8, Canada

5. Department of Molecular Genetics, University of Toronto, Toronto, ON M5S 1A8, Canada

Funder

Canadian Institutes of Health Research

Canada Research Chairs

Michael Smith Foundation for Health Research

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.1c00428

Reference16 articles.

1. Small-Molecule Inhibition of HIV pre-mRNA Splicing as a Novel Antiretroviral Therapy to Overcome Drug Resistance

2. A Parallel Synthesis Approach to the Identification of Novel Diheteroarylamide-Based Compounds Blocking HIV Replication: Potential Inhibitors of HIV-1 Pre-mRNA Alternative Splicing

3. Modulation of the splicing regulatory function of SRSF10 by a novel compound that impairs HIV-1 replication

4. Characterization of novel inhibitors of HIV-1 replication that function via alteration of viral RNA processing and rev function

5. Chemistry and Structure–Activity Relationships of Leukotriene Receptor Antagonists

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