Structure–Activity Relationship of Anti-<i>Mycobacterium abscessus</i> Piperidine-4-carboxamides, a New Class of NBTI DNA Gyrase Inhibitors-Reference-Cited by-同舟云学术

Structure–Activity Relationship of Anti-Mycobacterium abscessus Piperidine-4-carboxamides, a New Class of NBTI DNA Gyrase Inhibitors

Published:2022-02-28 Issue:3 Volume:13 Page:417-427
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Beuchel Andreas¹,Robaa Dina¹,Negatu Dereje A.²³,Madani Abdeldjalil²,Alvarez Nadine²,Zimmerman Matthew D.²,Richter Adrian¹^ORCID,Mann Lea¹,Hoenke Sophie⁴,Csuk René⁴^ORCID,Dick Thomas²⁵⁶,Imming Peter¹^ORCID

Affiliation:

1. Institut für Pharmazie, Martin-Luther-Universität Halle−Wittenberg, Halle, Germany, Kurt−Mothes−Str. 3, 06120 Halle (Saale), Germany

2. Center for Discovery and Innovation, Hackensack Meridian Health, Nutley, New Jersey 07110, United States

3. Center for Innovative Drug Development and Therapeutic Trials for Africa (CDT-Africa), Addis Ababa University, Addis Ababa 1000, Ethiopia

4. Institut für Chemie, Martin-Luther-University Halle−Wittenberg, Kurt−Mothes−Str. 2, 06120 Halle (Saale), Germany

5. Department of Medical Sciences, Hackensack Meridian School of Medicine, Nutley, New Jersey 07110, United States

6. Department of Microbiology and Immunology, Georgetown University, Washington, D.C. 20057, United States

Funder

National Institute of Allergy and Infectious Diseases

Deutsche Forschungsgemeinschaft

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.1c00549

Reference35 articles.

1. The Rise of Non-Tuberculosis Mycobacterial Lung Disease

2. The geographic diversity of nontuberculous mycobacteria isolated from pulmonary samples: an NTM-NET collaborative study

3. Failure to Recognize Nontuberculous Mycobacteria Leads to Misdiagnosis of Chronic Pulmonary Tuberculosis

4. DNA Topoisomerase Inhibitors: Trapping a DNA-Cleaving Machine in Motion

5. Mycobacterium tuberculosis Gyrase Inhibitors as a New Class of Antitubercular Drugs

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