GPBAR1 Activation by C6-Substituted Hyodeoxycholane Analogues Protect against Colitis-Reference-Cited by-同舟云学术

GPBAR1 Activation by C6-Substituted Hyodeoxycholane Analogues Protect against Colitis

Published:2020-03-02 Issue:5 Volume:11 Page:818-824
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Marino Simona De¹^ORCID,Finamore Claudia¹,Biagioli Michele²,Carino Adriana²,Marchianò Silvia²,Roselli Rosalinda¹,Giorgio Cristina Di²,Bordoni Martina²,Di Leva Francesco Saverio¹,Novellino Ettore¹^ORCID,Cassiano Chiara¹,Limongelli Vittorio¹³^ORCID,Zampella Angela¹^ORCID,Festa Carmen¹^ORCID,Fiorucci Stefano²

Affiliation:

1. Department of Pharmacy, University of Naples “Federico II”, Via D. Montesano 49, 80131 Naples, Italy

2. Department of Surgery and Biomedical Sciences, Nuova Facoltà di Medicina, Perugia CH-6900, Italy

3. Faculty of Biomedical Sciences, Institute of Computational Science, Center for Computational Medicine in Cardiology, Università della Svizzera italiana (USI), Via G. Buffi 13, CH-6900 Lugano, Switzerland

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.9b00636

Reference30 articles.

1. T-Cell Trafficking and Anti-Adhesion Strategies in Inflammatory Bowel Disease: Current and Future Prospects

2. Identification of membrane-type receptor for bile acids (M-BAR)

3. Bile acids induce energy expenditure by promoting intracellular thyroid hormone activation

4. Chemistry and Pharmacology of GPBAR1 and FXR Selective Agonists, Dual Agonists, and Antagonists

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