Development of a Water-Soluble Indolylmaleimide Derivative IM-93 Showing Dual Inhibition of Ferroptosis and NETosis

Author:

Dodo Kosuke123ORCID,Kuboki Erika4,Shimizu Tadashi13,Imamura Ryu5,Magarisawa Megumi4,Takahashi Masahiro3,Tokuhiro Takuto4,Yotsumoto Satoshi4,Asano Kenichi4,Nakao Shuhei1,Terayama Naoki1,Suda Takashi5,Tanaka Masato4,Sodeoka Mikiko123ORCID

Affiliation:

1. Synthetic Organic Chemistry Laboratory, RIKEN Cluster for Pioneering Research, 2-1, Hirosawa, Wako-shi, Saitama 351-0198, Japan

2. Sodeoka Live Cell Chemistry Project, ERATO, JST, 2-1, Hirosawa, Wako-shi, Saitama 351-0198, Japan

3. Institute of Multidisciplinary Research for Advanced Materials (IMRAM), Tohoku University, 2-1-1, Katahira, Aoba, Sendai, Miyagi 980-8577, Japan

4. Laboratory of Immune Regulation, School of Life Sciences, Tokyo University of Pharmacy and Life Sciences, 1432-1 Horinouchi, Hachiouji, Tokyo 192-0392, Japan

5. Division of Immunology and Molecular Biology, Cancer Research Institute, Kanazawa University, Kakuma-machi, Kanazawa, Ishikawa 920-1192, Japan

Funder

Naito Foundation

Takeda Science Foundation

Ministry of Education, Culture, Sports, Science and Technology

RIKEN

Japan Agency for Medical Research and Development

Japan Society for the Promotion of Science

Uehara Memorial Foundation

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

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