5,6-Dihydroxypyrimidine Scaffold to Target HIV-1 Nucleocapsid Protein

Author:

Malancona Savina1ORCID,Mori Mattia2ORCID,Fezzardi Paola1,Santoriello Marisabella1,Basta Andreina1,Nibbio Martina1,Kovalenko Lesia3,Speziale Roberto1,Battista Maria Rosaria1,Cellucci Antonella1,Gennari Nadia1,Monteagudo Edith1,Di Marco Annalise1,Giannini Alessia4,Sharma Rajhans3,Pires Manuel3,Real Eleonore3ORCID,Zazzi Maurizio4,Dasso Lang Maria Chiara2,De Forni Davide5,Saladini Francesco4,Mely Yves3ORCID,Summa Vincenzo1,Harper Steven1,Botta Maurizio2ORCID

Affiliation:

1. IRBM S.p.A., Via Pontina Km 30.600, 00071 Pomezia, Rome, Italy

2. Department of Biotechnology, Chemistry and Pharmacy, University of Siena, via Aldo Moro 2, 53100 Siena, Italy

3. Laboratoire de Bioimagerie et Pathologies, UMR 7021 CNRS, Faculté de Pharmacie, Université de Strasbourg, 74 Route du Rhin, 67401 Illkirch, France

4. Department of Medical Biotechnologies, University of Siena, Viale Mario Bracci, 16, 50100 Siena, Italy

5. ViroStatics S.r.l, Viale Umberto I 46, 07100 Sassari, Italy

Funder

Institut Universitaire de France

Seventh Framework Programme

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Reference33 articles.

1. UNAIDS. Global HIV & AIDS statistics - 2019 fact sheet; UNAIDS, 2020. https://www.unaids.org/en/resources/fact-sheet (accessed 2020-03-20).

2. AIDSinfo. Understanding HIV/AIDS-Fact Sheets; AIDSinfo, 2020. https://aidsinfo.nih.gov/understanding-hiv-aids (accessed on 2020-03-20).

3. Anti-HIV Drug Discovery and Development: Current Innovations and Future Trends

4. Retrospective on the all-in-one retroviral nucleocapsid protein

5. Role of HIV-1 nucleocapsid protein in HIV-1 reverse transcription

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