Pyrrolyl Pyrazoles as Non-Diketo Acid Inhibitors of the HIV-1 Ribonuclease H Function of Reverse Transcriptase-Reference-Cited by-同舟云学术

Pyrrolyl Pyrazoles as Non-Diketo Acid Inhibitors of the HIV-1 Ribonuclease H Function of Reverse Transcriptase

Published:2020-03-05 Issue:5 Volume:11 Page:798-805
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Messore Antonella¹,Corona Angela²^ORCID,Madia Valentina Noemi¹,Saccoliti Francesco¹,Tudino Valeria¹,De Leo Alessandro¹,Scipione Luigi¹,De Vita Daniela¹,Amendola Giorgio³^ORCID,Di Maro Salvatore³^ORCID,Novellino Ettore⁴^ORCID,Cosconati Sandro³^ORCID,Métifiot Mathieu⁵,Andreola Marie-Line⁵,Valenti Piera⁶,Esposito Francesca²,Grandi Nicole²,Tramontano Enzo²^ORCID,Costi Roberta¹^ORCID,Di Santo Roberto¹^ORCID

Affiliation:

1. Dipartimento di Chimica e Tecnologie del Farmaco, Istituto Pasteur-Fondazione Cenci Bolognetti, “Sapienza” Università di Roma, p.le Aldo Moro 5, I-00185 Roma, Italy

2. Department of Life and Environmental Sciences, University of Cagliari, Cittadella Universitaria di Monserrato, SS554-09042 Monserrato (CA), Italy

3. DiSTABiF, University of Campania “Luigi Vanvitelli”, Via Vivaldi 43, 81100 Caserta, Italy

4. Department of Pharmacy, University Federico II of Naples, Via D. Montesano 49, 80131 Naples, Italy

5. Laboratoire MFP, UMR 5234, CNRS, Université de Bordeaux, 146 rue Léo Saignat, 33076 Bordeaux cedex, France

6. Department of Public Health and Infectious Diseases, “Sapienza” University of Rome, p.le Aldo Moro 5, I-00185 Rome, Italy

Funder

Sapienza Universit? di Roma

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

http://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.9b00617

Reference29 articles.

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