Discovery of Potent and Selective 7-Azaindole Isoindolinone-Based PI3Kγ Inhibitors-Reference-Cited by-同舟云学术

Discovery of Potent and Selective 7-Azaindole Isoindolinone-Based PI3Kγ Inhibitors

Published:2020-09-24 Issue:11 Volume:11 Page:2244-2252
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Miles Dillon H.¹,Yan Xuelei¹,Thomas-Tran Rhiannon¹,Fournier Jeremy¹,Sharif Ehesan U.¹^ORCID,Drew Samuel L.¹,Mata Guillaume¹^ORCID,Lawson Kenneth V.¹^ORCID,Ginn Elaine¹,Wong Kent¹,Soni Divyank¹,Dhanota Puja¹,Shaqfeh Stefan G.¹,Meleza Cesar¹,Chen Ada¹,Pham Amber T.¹,Park Timothy¹,Swinarski Debbie¹,Banuelos Jesus¹,Schindler Ulrike¹,Walters Matthew J.¹,Walker Nigel P.¹,Zhao Xiaoning¹,Young Stephen W.¹,Chen Jie¹^ORCID,Jin Lixia¹,Leleti Manmohan Reddy¹,Powers Jay P.¹,Jeffrey Jenna L.¹^ORCID

Affiliation:

1. Arcus Biosciences, Inc., Hayward, California 94545, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.0c00387

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