Discovery of Novel Nonpeptidic PAR2 Ligands-Reference-Cited by-同舟云学术

Discovery of Novel Nonpeptidic PAR2 Ligands

Published:2020-05-22 Issue:6 Volume:11 Page:1316-1323
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Klösel Ilona¹,Schmidt Maximilian F.¹,Kaindl Jonas¹,Hübner Harald¹,Weikert Dorothee¹,Gmeiner Peter¹^ORCID

Affiliation:

1. Department of Chemistry and Pharmacy, Medicinal Chemistry, Friedrich-Alexander University Erlangen-Nürnberg (FAU), Nikolaus-Fiebiger-Str. 10, 91058 Erlangen, Germany

Funder

Elitenetzwerk Bayern

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.0c00154

Reference39 articles.

1. The structure and function of G-protein-coupled receptors

2. Protease-Activated Receptors: Contribution to Physiology and Disease

3. Structure, function and pathophysiology of protease activated receptors

4. Essential role for proteinase-activated receptor-2 in arthritis

5. Protease-activated receptor-2 in endosomes signals persistent pain of irritable bowel syndrome

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