Covalent Inhibition of Wild-Type HIV-1 Reverse Transcriptase Using a Fluorosulfate Warhead-Reference-Cited by-同舟云学术

Covalent Inhibition of Wild-Type HIV-1 Reverse Transcriptase Using a Fluorosulfate Warhead

Published:2021-01-06 Issue:2 Volume:12 Page:249-255
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Ippolito Joseph A.¹²,Niu Haichan¹,Bertoletti Nicole²^ORCID,Carter Zachary J.¹,Jin Shengyan²,Spasov Krasimir A.²,Cisneros José A.¹,Valhondo Margarita¹,Cutrona Kara J.¹,Anderson Karen S.²³^ORCID,Jorgensen William L.¹^ORCID

Affiliation:

1. Department of Chemistry, Yale University, New Haven, Connecticut 06520-8107, United States,

2. Department of Pharmacology, Yale University School of Medicine, New Haven, Connecticut 06520-8066, United States

3. Department of Molecular Biophysics and Biochemistry, Yale University School of Medicine, New Haven, Connecticut 06520-8066, United States

Funder

National Institute of Allergy and Infectious Diseases

National Institute of General Medical Sciences

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.0c00612

Reference29 articles.

1. Global, regional, and national incidence, prevalence, and mortality of HIV, 1980–2017, and forecasts to 2030, for 195 countries and territories: a systematic analysis for the Global Burden of Diseases, Injuries, and Risk Factors Study 2017

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3. Single-Tablet Regimens for the Treatment of HIV-1 Infection

4. Current and emerging non-nucleoside reverse transcriptase inhibitors (NNRTIs) for HIV-1 treatment

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