Discovery of Potent and Orally Bioavailable Small Molecule Antagonists of Toll-like Receptors 7/8/9 (TLR7/8/9)
Author:
Affiliation:
1. Bristol Myers Squibb Research and Development, P.O. Box 4000, Princeton, New Jersey 08543, United States
2. The Biocon Bristol Myers Squibb Research Center (BBRC), Bangalore 560099, India
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Drug Discovery,Biochemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.0c00264
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1. Sensors of the innate immune system: their mode of action
2. The history of Toll-like receptors — redefining innate immunity
3. Immunologically Active Autoantigens: The Role of Toll-Like Receptors in the Development of Chronic Inflammatory Disease
4. Species-Specific Recognition of Single-Stranded RNA via Toll-like Receptor 7 and 8
5. A Tlr7 translocation accelerates systemic autoimmunity in murine lupus
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