Development of a Raltegravir-based Photoaffinity-Labeled Probe for Human Immunodeficiency Virus-1 Integrase Capture-Reference-Cited by-同舟云学术

Development of a Raltegravir-based Photoaffinity-Labeled Probe for Human Immunodeficiency Virus-1 Integrase Capture

Published:2020-04-28 Issue:10 Volume:11 Page:1986-1992
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Pala Nicolino¹,Esposito Francesca²,Tramontano Enzo²^ORCID,Singh Pankaj Kumar¹,Sanna Vanna³^ORCID,Carcelli Mauro⁴^ORCID,Haigh Lisa D.⁵,Satta Sandro⁶⁷,Sechi Mario¹^ORCID

Affiliation:

1. Department of Chemistry and Pharmacy, Laboratory of Drug Design and Nanomedicine, University of Sassari, Sassari 07100, Italy

2. Department of Life and Environmental Sciences, University of Cagliari, Cagliari 09042, Italy

3. Nanomater s.r.l., c/o Porto Conte Ricerche, Alghero 07041, Italy

4. Department of Chemistry, Life Sciences and Environmental Sustainability, University of Parma, Parma 43124, Italy

5. Department of Chemistry, Imperial College London, London W12 0BZ, United Kingdom

6. Centre for Pharmacology & Therapeutics, Department of Medicine, Imperial College London, London W12 0NN, United Kingdom

7. Department of Medicine, David Geffen School of Medicine, University of California, Los Angeles, California 90095, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

http://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.0c00009

Reference36 articles.

1. New Paradigms in Drug Design and Discovery

2. Principles of early drug discovery

3. X-ray crystallography: assessment and validation of protein–small molecule complexes for drug discovery

4. Photoaffinity labeling in target- and binding-site identification

5. Using photolabile ligands in drug discovery and development

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