Covalent <i>S</i>-Adenosylhomocysteine-Based DNA Methyltransferase 2 Inhibitors with a New Type of Aryl Warhead-Reference-Cited by-同舟云学术

Covalent S-Adenosylhomocysteine-Based DNA Methyltransferase 2 Inhibitors with a New Type of Aryl Warhead

Published:2023-05-09 Issue:6 Volume:14 Page:777-787
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Schwickert Marvin¹^ORCID,Zimmermann Robert A.¹^ORCID,Habeck Tanja²,Hoba Sabrina N.¹,Nidoieva Zarina¹^ORCID,Fischer Tim R.¹,Stark Martin M.¹,Kersten Christian¹^ORCID,Lermyte Frederik²,Helm Mark¹^ORCID,Schirmeister Tanja¹

Affiliation:

1. Institute of Pharmaceutical and Biomedical Sciences, Johannes Gutenberg University Mainz, Staudinger Weg 5, D-55128 Mainz, Germany

2. Technical University of Darmstadt, Alarich-Weiss-Strasse 4, D-64287 Darmstadt, Germany

Funder

Deutsche Forschungsgemeinschaft

Fonds der Chemischen Industrie

Hessisches Ministerium f?r Wissenschaft und Kunst

Volkswagen Foundation

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.3c00062

Reference21 articles.

1. The RNA modification landscape in human disease

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