Discovery and Pharmacology of a Novel Somatostatin Subtype 5 (SSTR5) Antagonist: Synergy with DPP-4 Inhibition
Author:
Affiliation:
1. Merck & Co., Inc., Kenilworth, New Jersey 07033, United States
Funder
Merck
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Drug Discovery,Biochemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.8b00305
Reference22 articles.
1. Advances in understanding neuronal somatostatin receptors
2. All Five Cloned Human Somatostatin Receptors (hSSTR1-5) Are Functionally Coupled to Adenylyl Cyclase
3. Molecular Biology of Somatostatin Receptors*
4. Somatostatin-28 regulates GLP-1 secretion via somatostatin receptor subtype 5 in rat intestinal cultures
5. Expression and Distribution of Somatostatin Receptor Subtypes in the Pancreatic Islets of Mice and Rats
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