Tuning the Dual Inhibition of Carbonic Anhydrase and Cyclooxygenase by Dihydrothiazole Benzensulfonamides-Reference-Cited by-同舟云学术

Tuning the Dual Inhibition of Carbonic Anhydrase and Cyclooxygenase by Dihydrothiazole Benzensulfonamides

Published:2018-09-17 Issue:10 Volume:9 Page:1045-1050
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Meleddu Rita¹,Distinto Simona¹^ORCID,Cottiglia Filippo¹^ORCID,Angius Rossella²,Gaspari Marco³^ORCID,Taverna Domenico³,Melis Claudia¹,Angeli Andrea⁴,Bianco Giulia¹,Deplano Serenella¹,Fois Benedetta¹,Del Prete Sonia⁵,Capasso Clemente⁵,Alcaro Stefano⁶,Ortuso Francesco⁶^ORCID,Yanez Matilde⁷,Supuran Claudiu T.⁴^ORCID,Maccioni Elias¹

Affiliation:

1. Department of Life and Environmental Sciences, University of Cagliari, Via Ospedale 72, 09124 Cagliari, Italy

2. Laboratorio NMR e Tecnologie Bioanalitiche, Sardegna Ricerche, 09010 Pula, Cagliari, Italy

3. Department of Experimental and Clinical Medicine, “Magna Græcia” University of Catanzaro, Campus ‘S. Venuta’, Viale Europa, 88100 Catanzaro, Italy

4. Dipartimento NEUROFARBA, Sezione di Scienze Farmaceutiche, Università degli Studi di Firenze, Sesto Fiorentino, Florence, Italy

5. Istituto di Bioscienze e Biorisorse, CNR, Via Pietro Castellino 111, 80131, Napoli, Italy

6. Dipartimento di Scienze della Salute, Università Magna Graecia di Catanzaro, Campus ‘S. Venuta’, Viale Europa, 88100 Catanzaro, Italy

7. Department of Pharmacology, Faculty of Pharmacy, University of Santiago de Compostela (USC), Santiago de Compostela, Spain

Funder

European Cooperation in Science and Technology

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.8b00352

Reference51 articles.

1. Dual Cyclooxygenase and Carbonic Anhydrase Inhibition by Nonsteroidal Anti-Inflammatory Drugs for the Treatment of Cancer

2. Carbonic anhydrase/COX-2 inhibitors in the treatment of various diseases

3. COX-2 Selective Inhibitors, Carbonic Anhydrase Inhibition and Anticancer Properties of Sulfonamides Belonging to This Class of Pharmacological Agents

4. Drug Design Studies of the Novel Antitumor Targets Carbonic Anhydrase IX and XII

5. Evolution and distribution of the carbonic anhydrase gene families

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