Imidazo[2,1-b]benzothiazol Derivatives as Potential Allosteric Inhibitors of the Glucocorticoid Receptor

Author:

Christodoulou Michael S.1ORCID,Dapiaggi Federico2,Ghiringhelli Francesca2,Pieraccini Stefano23,Sironi Maurizio23,Lucafò Marianna4,Curci Debora5,Decorti Giuliana46,Stocco Gabriele7,Chirumamilla Chandra Sekhar8,Vanden Berghe Wim8ORCID,Balaguer Patrick9,Michel Benoît Y.10,Burger Alain10,Beccalli Egle M.1,Passarella Daniele2ORCID,Martinet Nadine10

Affiliation:

1. DISFARM, Sezione di Chimica Generale e Organica “A. Marchesini”, Università degli Studi di Milano, Via Venezian 21, 20133 Milano, Italy

2. Department of Chemistry, Università degli Studi di Milano, Via Golgi 19, 20133 Milano Italy

3. Istituto di Scienze e Tecnologie Molecolari (INSTM), CNR, and INSTM, UdR Milano, Via Golgi 19, 20133 Milano, Italy

4. Department of Medicine, Surgery and Health Sciences, University of Trieste, 34127 Trieste, Italy

5. PhD School in Reproduction and Developmental Sciences, University of Trieste, 34127 Trieste, Italy

6. Institute for Maternal and Child Health - IRCCS “Burlo Garofolo”, 34127 Trieste, Italy

7. Department of Life Sciences, University of Trieste, 34127 Trieste, Italy

8. Laboratory of Protein Chemistry, Proteomics and Epigenetic Signalling, Department of Biomedical Sciences, University of Antwerp (UA), 2000 Antwerpen, Belgium

9. IRCM, INSERM U1194, Université Montpellier, ICM, 208 rue des Apothicaires, F-34298 Montpellier, France

10. Université Côte d’Azur, CNRS, Institut de Chimie de Nice, UMR 7272, Parc Valrose, 06108 Nice Cedex 2, France

Funder

European Cooperation in Science and Technology

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

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