A Combination of Docking/Dynamics Simulations and Pharmacophoric Modeling To Discover New Dual c-Src/Abl Kinase Inhibitors-Reference-Cited by-同舟云学术

A Combination of Docking/Dynamics Simulations and Pharmacophoric Modeling To Discover New Dual c-Src/Abl Kinase Inhibitors

Published:2006-05-06 Issue:11 Volume:49 Page:3278-3286
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Manetti Fabrizio¹,Locatelli Giada A.¹,Maga Giovanni¹,Schenone Silvia¹,Modugno Michele¹,Forli Stefano¹,Corelli Federico¹,Botta Maurizio¹

Affiliation:

1. Dipartimento Farmaco Chimico Tecnologico, Università degli Studi di Siena, Via Alcide de Gasperi 2, I-53100, Siena, Italy, Istituto di Genetica Molecolare, IGM-CNR, Via Abbiategrasso 207, I-27100, Pavia, Italy, and Dipartimento di Scienze Farmaceutiche, Università degli Studi di Genova, Viale Benedetto XV 3, I-16132, Genova, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm060236z

Reference32 articles.

1. The hunting of the Src

2. v-SRC'S hold over actin and cell adhesions

3. Selected glimpses into the activation and function of Src kinase

4. Expression of pp60c-src in human small cell and non-small cell lung carcinomas

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