Structure–Activity Relationship Studies on Isoindoline Inhibitors of Dipeptidyl Peptidases 8 and 9 (DPP8, DPP9): Is DPP8-Selectivity an Attainable Goal?-Reference-Cited by-同舟云学术

Structure–Activity Relationship Studies on Isoindoline Inhibitors of Dipeptidyl Peptidases 8 and 9 (DPP8, DPP9): Is DPP8-Selectivity an Attainable Goal?

Published:2011-08-02 Issue:16 Volume:54 Page:5737-5746
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Van Goethem Sebastiaan¹,Matheeussen Veerle²,Joossens Jurgen¹,Lambeir Anne-Marie²,Chen Xin³,De Meester Ingrid²,Haemers Achiel¹,Augustyns Koen¹,Van der Veken Pieter¹

Affiliation:

1. Laboratory of Medicinal Chemistry, Department of Pharmaceutical Sciences, University of Antwerp (UA), Universiteitsplein 1, B-2610 Wilrijk, Antwerp, Belgium

2. Laboratory of Medical Biochemistry, Department of Pharmaceutical Sciences, University of Antwerp (UA), Universiteitsplein 1, B-2610 Antwerp, Belgium

3. Division of Biotechnology and Pharmaceutical Research, National Health Research Institutes, Zhu Nan, Miaoli 350, Taiwan, ROC

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm200383j

Reference48 articles.

1. The dipeptidyl peptidase IV family in cancer and cell biology

2. The Therapeutic Potential of Inhibitors of Dipeptidyl Peptidase IV (DPP IV) and Related Proline-Specific Dipeptidyl Aminopeptidases

3. Prolyl Peptidases Related to Dipeptidyl Peptidase IV: Potential of Specific Inhibitors in Drug Discovery.

4. Dipeptidyl peptidase IV activity and/or structure homologues (DASH) and their substrates in cancer

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