Refinement of the Benzodiazepine Receptor Site Topology by Structure−Activity Relationships of New N-(Heteroarylmethyl)indol-3-ylglyoxylamides-Reference-Cited by-同舟云学术

Refinement of the Benzodiazepine Receptor Site Topology by Structure−Activity Relationships of New N-(Heteroarylmethyl)indol-3-ylglyoxylamides

Published:2006-03-30 Issue:8 Volume:49 Page:2489-2495
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Primofiore Giampaolo¹,Da Settimo Federico¹,Marini Anna Maria¹,Taliani Sabrina¹,La Motta Concettina¹,Simorini Francesca¹,Novellino Ettore¹,Greco Giovanni¹,Cosimelli Barbara¹,Ehlardo Marina¹,Sala Annalisa¹,Besnard François¹,Montali Marina¹,Martini Claudia¹

Affiliation:

1. Dipartimento di Scienze Farmaceutiche, Università di Pisa, Via Bonanno 6, 56126 Pisa, Italy, Dipartimento di Chimica Farmaceutica e Tossicologica, Università di Napoli “Federico II”, Via Domenico Montesano, 49, 80131 Napoli, Italy, Department of Molecular and Functional Genomics, Synthélabo, 10 rue des Carrières, 92500 Rueil-Malmaison, France, and Dipartimento di Psichiatria, Neurobiologia, Farmacologia e Biotecnologie, Università di Pisa, Via Bonanno 6, 56126 Pisa, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0511841

Reference41 articles.

1. GABA-Activated Ligand Gated Ion Channels: Medicinal Chemistry and Molecular Biology

2. An update on GABAA receptors

3. Mapping of the Benzodiazepine Recognition Site on GABA-A Receptors

4. Subunit Composition, Distribution and Function of GABA-A Receptor Subtypes

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